, , ; "10.1016/j.bmcl.2016.07.081"^^; ; ; "27524313"^^; "René O, Fauber BP, Barnard A, Chapman K, Deng Y, Eidenschenk C, Everett C, Gobbi A, Johnson AR, La H, Norman M, Salmon G, Summerhill S, Wong H.: Discovery of oxa-sultams as RORc inverse agonists showing reduced lipophilicity, improved selectivity and favorable ADME properties. Bioorg Med Chem Lett, Volume 26 (18), 2016"^^ . . . . .